Peptide Active Data Details
Basic Peptide Information
DICL ID
DICL_Pep_00500
Ion Channel
Voltage-gated potassium channel subfamily KQT member 1
Peptide Function
Inhibitor
Gene Name
KCNQ1
Activity Data (nM)
IC50
5000 nM
Ki
Not available
EC50
Not available
Kd
Not available
Biologically Active
Not specified
Sequence Information
Peptide Sequence
CNCKAPETALCARRCQQH
Peptide UniProt Accession
UniParc
UPI0000035420
Peptide Synonyms/Alias
[Apamin; Apamine; UNII-X644P85KUR; EINECS 246-182-7; C79H131N31O24S4; Ro 23-6721; X644P85KUR; NS00075519; Q417260]
Peptide Species
Apis mellifera (Honeybee)
Peptide Name
Apamin
CAS Number
24345-16-2
Experimental Conditions
pH
pH 7.4
Holding Potential (mV)
−90 mV
Temperature
18–22 °C
Test Method
Patch-clamping
Test Species
Xenopus laevis oocyte
Binding Information
Binding Site
Not specified
Binding Site Residue
Not specified
Ion Channel Information
Gene Abbreviation (ABB)
VGKCs
Ion Channel UniProt Accession
Source Organism
Rattus norvegicus (Rat)
References & Disease Information
Disease
Not specified
PubChem CID
URL
Not available
PMID
Patent
Not available